SCHEMBL28865411

SCHEMBL28865411

Nc1nccc(Nc2ccc(CCCF)cc2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 11/20 0.56
BCL6 P41182 1/20 0.56
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA6 P23280 1/20 0.52
CA5A P35218 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52
CA5B Q9Y2D0 1/20 0.52
KCNH2 Q12809 1/20 0.50
SCN9A Q15858 1/20 0.50
HRH3 Q9Y5N1 1/20 0.47
ROCK2 O75116 1/20 0.46
PRKACA P17612 1/20 0.46
PRKCD Q05655 1/20 0.46
DYRK1A Q13627 1/20 0.46
CDC42BPA Q5VT25 1/20 0.46
HTR3E A5X5Y0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12346577 0.87 ROCK1 (0.61) ROCK1BCL6CA12CA1CA2
SCHEMBL12968977 0.79 ROCK1 (0.63) ROCK1BCL6CA12CA1CA2
SCHEMBL31336991 0.77 ROCK1 (0.69) ROCK1BCL6CA12CA1CA2
SCHEMBL28247390 0.77 ROCK1 (0.59) ROCK1BCL6CA12CA1CA2
SCHEMBL1935543 0.76 ROCK1 (0.58) ROCK1BCL6CA12CA1CA2
SCHEMBL12968976 0.75 ROCK1 (0.65) ROCK1BCL6CA12CA1CA2
Hydrochloric Acid SCHEMBL12813104 0.74 ROCK1 (0.63) ROCK1BCL6CA12CA1CA2
SCHEMBL31337029 0.73 SCN9A (0.82) ROCK1BCL6CA12CA1CA2
SCHEMBL13963140 0.73 ROCK1 (0.69) ROCK1BCL6CA12CA1CA2
SCHEMBL31337079 0.73 ROCK1 (0.69) ROCK1BCL6CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105348203-B Inhibit the composition and method of JAK approach 里格尔药品股份有限公司 2018-09-18 CN disclosed