SCHEMBL288656

SCHEMBL288656

COc1cc(CN2C(=O)CCC2C(=O)N[C@H](Cc2ccccc2)C(=O)C(N)=O)cc(OC)c1

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 11/20 0.71
ITGB1 P05556 9/20 0.54
ITGA4 P13612 9/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287861 1.00 CAPN1 (0.71) CAPN1ITGB1ITGA4
SCHEMBL298845 1.00 CAPN1 (0.71) CAPN1ITGB1ITGA4
SCHEMBL289791 1.00 CAPN1 (0.71) CAPN1ITGB1ITGA4
SCHEMBL299450 0.94 CAPN1 (0.70) CAPN1ITGB1ITGA4
SCHEMBL288173 0.94 CAPN1 (0.70) CAPN1ITGB1ITGA4
SCHEMBL289316 0.94 CAPN1 (0.70) CAPN1ITGB1ITGA4
SCHEMBL1612436 0.89 CAPN1 (0.88) CAPN1ITGB1ITGA4
SCHEMBL288617 0.89 CAPN1 (0.88) CAPN1ITGB1ITGA4
SCHEMBL288910 0.89 CAPN1 (0.88) CAPN1ITGB1ITGA4
SCHEMBL288113 0.87 CAPN1 (0.74) CAPN1ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427429-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS Abbott GmbH & Co. KG (DE) 2012-03-14 EP disclosed
WO-2010128102-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS ABBOTT GMBH & CO. KG (DE) 2010-11-11 WO disclosed