SCHEMBL28867039

SCHEMBL28867039

Ic1ccc2cn(-c3ccnc4[nH]ccc34)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 7/20 0.48
AKT2 P31751 1/20 0.40
NUDT1 P36639 5/20 0.39
AXL P30530 1/20 0.37
PBK Q96KB5 1/20 0.37
CCNK O75909 2/20 0.35
CDK12 Q9NYV4 2/20 0.35
AURKB Q96GD4 2/20 0.34
AURKA O14965 1/20 0.34
INCENP Q9NQS7 1/20 0.34
TPX2 Q9ULW0 1/20 0.34
GRM4 Q14833 1/20 0.34
RHEB Q15382 1/20 0.34
IKBKB O14920 1/20 0.34
CHUK O15111 1/20 0.34
DAPK3 O43293 1/20 0.34
JAK2 O60674 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
PAK4 O96013 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29941811 1.00 PRKCI (0.48) PRKCIAKT2NUDT1AXLPBK
SCHEMBL100370 0.82 PRKCI (0.52) PRKCIAKT2NUDT1AXLPBK
SCHEMBL100896 0.80 MEN1 (0.52) PRKCIAKT2NUDT1JAK2JAK3
SCHEMBL29540654 0.80 MEN1 (0.52) PRKCIAKT2NUDT1JAK2JAK3
Trifluoroacetic Acid SCHEMBL4092152 0.73 KMT2A (0.47) PRKCIPBKAURKBAURKARHEB
SCHEMBL28867033 0.73 MAP3K14 (0.47) PRKCIAKT2NUDT1PBKPAK4
SCHEMBL100232 0.73 PRKCI (0.44) PRKCIAKT2NUDT1JAK2JAK3
SCHEMBL29940967 0.72 PRKCI (0.45) PRKCIAKT2NUDT1AXLPBK
SCHEMBL28867026 0.72 PRKCI (0.45) PRKCIAKT2NUDT1AXLPBK
Trifluoroacetic Acid SCHEMBL4086134 0.72 PRKCI (0.43) PRKCIAKT2NUDT1PBKAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115215861-B Aromatic heterocycle substituted alkyne compound and preparation method and application thereof 上海翊石医药科技有限公司 2024-03-15 CN disclosed
CN-115215861-A Aromatic heterocycle substituted alkyne compound and preparation method and application thereof 上海翊石医药科技有限公司 2022-10-21 CN disclosed