SCHEMBL288718

SCHEMBL288718

N[C@H](CC(=O)O)Cc1ccccn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRA P18433 1/20 0.58
DPP4 P27487 2/20 0.56
GRIN2D O15399 1/20 0.56
GRIN3B O60391 1/20 0.56
GRIN1 Q05586 1/20 0.56
GRIN2A Q12879 1/20 0.56
GRIN2B Q13224 1/20 0.56
GRIN2C Q14957 1/20 0.56
GRIN3A Q8TCU5 1/20 0.56
FDPS P14324 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 1/20 0.46
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
POLB P06746 1/20 0.42
HRH1 P35367 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532234 0.84 SMN1; SMN2 (0.51) PTPRADPP4GRIN2DGRIN3BGRIN1
SCHEMBL4301092 0.82 MAPK1 (0.56) PTPRADPP4GRIN2DGRIN3BGRIN1
SCHEMBL6997949 0.82 GRIN2D (0.66) PTPRADPP4GRIN2DGRIN3BGRIN1
SCHEMBL8507957 0.80 KDM4E (0.57) PTPRASMN1; SMN2CYP1A2CYP2D6MAPT
SCHEMBL8509020 0.80 PTPRA (0.51) PTPRADPP4GRIN2DGRIN3BGRIN1
SCHEMBL28378998 0.80 PTPRA (0.58) PTPRAGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL126508 0.79 PTPRA (0.67) PTPRADPP4GRIN2DGRIN3BGRIN1
SCHEMBL22409316 0.79 PTPRA (0.67) PTPRADPP4GRIN2DGRIN3BGRIN1
SCHEMBL29401000 0.79 PTPRA (0.67) PTPRADPP4GRIN2DGRIN3BGRIN1
SCHEMBL29805516 0.79 PTPRA (0.67) PTPRADPP4GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104284891-B Conformationally constrained, fully synthetic macrocyclic compounds 波利弗尔股份公司 2018-04-17 CN disclosed
EP-2427476-A1 BETA-HAIRPIN PEPTIDOMIMETICS HAVING CXCR4 ANTAGONIZING ACTIVITY Polyphor Ag (CH) 2012-03-14 EP disclosed
WO-2010127704-A1 BETA-HAIRPIN PEPTIDOMIMETICS HAVING CXCR4 ANTAGONIZING ACTIVITY POLYPHOR AG (CH) 2010-11-11 WO disclosed