SCHEMBL28876151

SCHEMBL28876151

O=C(NO)c1cccc(Nc2nc(Nc3ccc(N4CCCCC4)cc3)ncc2F)c1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.59
CCNT1 O60563 6/20 0.57
CCNE1 P24864 6/20 0.57
CDK2 P24941 6/20 0.57
CDK9 P50750 6/20 0.57
SYK P43405 2/20 0.56
GSK3A P49840 1/20 0.52
GSK3B P49841 1/20 0.52
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
FLT3 P36888 2/20 0.51
BTK Q06187 2/20 0.51
AURKA O14965 3/20 0.51
JAK2 O60674 1/20 0.50
AURKB Q96GD4 1/20 0.50
EGFR P00533 1/20 0.49
SCN9A Q15858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29463618 1.00 BRD4 (0.59) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL28714151 0.92 FLT3 (0.59) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL29514559 0.92 FLT3 (0.59) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL28876155 0.92 SYK (0.69) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL29463619 0.92 SYK (0.69) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL29463626 0.91 BRD4 (0.72) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL28876170 0.91 BRD4 (0.72) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL28876165 0.90 BRD4 (0.65) BRD4SYKGSK3AGSK3BHDAC3
SCHEMBL29463622 0.89 BRD4 (0.59) BRD4CCNT1CCNE1CDK2CDK9
SCHEMBL28876153 0.89 BRD4 (0.59) BRD4CCNT1CCNE1CDK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114230524-A (5-fluoro-2-anilinopyrimidin-4-yl) amino-N-hydroxybenzamide derivative and preparation method and application thereof 南通大学 2022-03-25 CN claimed
CN-114230524-A (5-fluoro-2-anilinopyrimidin-4-yl) amino-N-hydroxybenzamide derivative and preparation method and application thereof 南通大学 2022-03-25 CN disclosed