SCHEMBL28882004

SCHEMBL28882004

Cc1ccc(NC(=O)C=Cc2cccc(-c3cnc4[nH]ccc4c3)c2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 14/20 0.74
MMP1 P03956 2/20 0.55
MMP2 P08253 2/20 0.55
MMP9 P14780 2/20 0.55
CDK7 P50613 2/20 0.54
PLK4 O00444 1/20 0.54
DCLK1 O15075 1/20 0.54
ROCK2 O75116 1/20 0.54
PRKD3 O94806 1/20 0.54
MAP4K4 O95819 1/20 0.54
PAK4 O96013 1/20 0.54
CHEK2 O96017 1/20 0.54
INSR P06213 1/20 0.54
CDK1 P06493 1/20 0.54
FES P07332 1/20 0.54
ROS1 P08922 1/20 0.54
PDGFRB P09619 1/20 0.54
PDGFRA P16234 1/20 0.54
FER P16591 1/20 0.54
CDK2 P24941 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29883569 1.00 CDK8 (0.74) CDK8MMP1MMP2MMP9CDK7
SCHEMBL28882046 0.91 CDK8 (0.73) CDK8MMP1MMP2MMP9CDK7
SCHEMBL29883221 0.91 CDK8 (0.73) CDK8MMP1MMP2MMP9CDK7
SCHEMBL29883381 0.91 CDK8 (0.82) CDK8CDK7PLK4DCLK1ROCK2
SCHEMBL28882044 0.91 CDK8 (0.82) CDK8CDK7PLK4DCLK1ROCK2
SCHEMBL29883357 0.90 CDK8 (0.71) CDK8MMP1MMP2MMP9CDK7
SCHEMBL29883280 0.90 CDK8 (0.69) CDK8MMP1MMP2MMP9CDK7
SCHEMBL28882270 0.90 CDK8 (0.71) CDK8MMP1MMP2MMP9CDK7
SCHEMBL28958611 0.90 CDK8 (0.69) CDK8MMP1MMP2MMP9CDK7
SCHEMBL28882047 0.89 CDK8 (0.68) CDK8MMP1MMP2MMP9CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115141197-B 3-aromatic heterocycle substituted phenyl derivative and preparation method and application thereof 安徽医科大学 2024-03-26 CN disclosed
CN-115141197-A 3-aromatic heterocyclic substituted phenyl derivative and preparation method and application thereof 安徽医科大学 2022-10-04 CN disclosed