SCHEMBL28883255

SCHEMBL28883255

O=C(NCC(O)CCCO)c1cc2cc(-c3ccc(F)cc3)ccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 2/20 0.45
AKR1C3 P42330 1/20 0.43
DRD3 P35462 3/20 0.42
DRD4 P21917 2/20 0.42
RXFP1 Q9HBX9 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28882540 0.92 KDM4E (0.45) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL28882553 0.85 DRD4 (0.42) KDM4EALDH1A1AKR1C3DRD3DRD4
SCHEMBL28352944 0.82 HDAC3 (0.55) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL28352663 0.82 KDM4E (0.44) KDM4EALDH1A1AKR1C3DRD3DRD4
SCHEMBL28353184 0.82 KDM4E (0.41) HDAC3HDAC1KDM4EALDH1A1AKR1C3
SCHEMBL28352701 0.82 KDM4E (0.46) KDM4EALDH1A1AKR1C3DRD3DRD4
SCHEMBL28352871 0.81 GRIN2D (0.46) KDM4EALDH1A1AKR1C3DRD3DRD4
SCHEMBL20615447 0.81 KDM4E (0.46) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL20615824 0.81 KDM4E (0.46) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL28885809 0.81 KDM4E (0.46) HDAC3HDAC1HDAC4HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110770224-B Indole derivatives as efflux pump inhibitors 罗格斯新泽西州立大学 2022-11-18 CN disclosed
CN-110770224-A Indole derivatives as efflux pump inhibitors 罗格斯新泽西州立大学 2020-02-07 CN disclosed