SCHEMBL28896381

SCHEMBL28896381

CCOC(=O)NC(=S)N(CC(CNC(=O)OC(C)(C)C)OC(F)C(F)F)c1cc[nH]c1C(=O)OCC

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SERPINE1 P05121 1/20 0.32
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28896379 0.90 KDM4E (0.32) KDM4EMAPTTDP1NPSR1SERPINE1
SCHEMBL29211242 0.79 AAK1 (0.38) KDM4EMAPTTDP1NPSR1
SCHEMBL28896258 0.79 MAPT (0.36) KDM4EMAPTTDP1NPSR1SERPINE1
SCHEMBL28896529 0.77
SCHEMBL28896526 0.77 MAPT (0.30) MAPTNPSR1
SCHEMBL28896243 0.75 CA12 (0.32) KDM4ENPSR1
SCHEMBL28896569 0.74 CA12 (0.32)
SCHEMBL28896338 0.73 AAK1 (0.37) KDM4EMAPTTDP1NPSR1SYK
SCHEMBL28896343 0.73 AAK1 (0.37) KDM4EMAPTTDP1NPSR1SYK
SCHEMBL28896564 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403584-A 2-thio-2, 3-dihydropyrimidine-4-one derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-29 CN disclosed