SCHEMBL28898468

SCHEMBL28898468

CC(C)(C)OC(=O)n1c(CN(CCC(N)=O)C2CCCc3cccnc32)nc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.49
KCNH2 Q12809 2/20 0.45
CHRM2 P08172 1/20 0.43
CYP2D6 P10635 1/20 0.43
DRD2 P14416 1/20 0.43
OPRM1 P35372 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22894729 1.00 CXCR4 (0.49) CXCR4KCNH2CHRM2CYP2D6DRD2
SCHEMBL5050923 0.90 CXCR4 (0.53) CXCR4KCNH2CHRM2CYP2D6DRD2
SCHEMBL4828646 0.88 CXCR4 (0.50) CXCR4KCNH2CHRM2CYP2D6DRD2
SCHEMBL14303642 0.88 CXCR4 (0.52) CXCR4KCNH2CHRM2CYP2D6DRD2
SCHEMBL5054280 0.88 CXCR4 (0.54) CXCR4
SCHEMBL3375920 0.88 CXCR4 (0.49) CXCR4CYP2D6
SCHEMBL5057529 0.87 CXCR4 (0.58) CXCR4KCNH2CHRM2CYP2D6DRD2
SCHEMBL4713761 0.87 CXCR4 (0.48) CXCR4KCNH2CHRM2CYP2D6DRD2
SCHEMBL5054150 0.86 CXCR4 (0.46) CXCR4
SCHEMBL4716687 0.86 CXCR4 (0.50) CXCR4KCNH2CHRM2CYP2D6DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111655261-A Acyclic CXCR4 inhibitors and uses thereof X4 制药有限公司 2020-09-11 CN disclosed