SCHEMBL28902818

SCHEMBL28902818

CC(C)(C)OC(=O)Nc1nc2c(O)c(F)ccc2s1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LCK P06239 14/20 0.47
MAPT P10636 2/20 0.45
DYRK1A Q13627 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30231217 1.00 LCK (0.47) LCKMAPTDYRK1ANPC1RAB9A
SCHEMBL33525654 0.86 LCK (0.49) LCKMAPTNPC1RAB9A
SCHEMBL25382677 0.84 LCK (0.45) LCKMAPTNPC1RAB9A
SCHEMBL30231211 0.84 LCK (0.45) LCKMAPTNPC1RAB9A
SCHEMBL30237087 0.83 LCK (0.44) LCKMAPTDYRK1A
SCHEMBL28902830 0.83 LCK (0.44) LCKMAPTDYRK1A
SCHEMBL21901580 0.81 LCK (0.45) LCKDYRK1A
SCHEMBL21901426 0.81 LCK (0.46) LCK
SCHEMBL30064634 0.81 LCK (0.46) LCK
SCHEMBL30231276 0.80 LCK (0.42) LCKMAPTDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116390923-A Heterocyclic derivative and preparation method and application thereof 浙江海正药业股份有限公司 2023-07-04 CN disclosed
CN-115403575-A Heteroaromatic ring derivative and preparation method and application thereof 浙江海正药业股份有限公司 2022-11-29 CN disclosed
CN-115385912-A Pyrazinopyrazinoquinolinone derivatives, preparation method and medical application thereof 浙江海正药业股份有限公司 2022-11-25 CN disclosed