SCHEMBL28911784

SCHEMBL28911784

O=C(Nc1cnccc1OC(F)C(F)F)c1ccnc(NCc2cccc(F)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 16/20 0.48
GSK3A P49840 15/20 0.48
PIM1 P11309 5/20 0.43
CDK2 P24941 3/20 0.43
JAK2 O60674 2/20 0.43
CDK5 Q00535 2/20 0.43
PRKCQ Q04759 2/20 0.43
AURKB Q96GD4 2/20 0.43
TYK2 P29597 1/20 0.43
SYK P43405 1/20 0.43
HDAC1 Q13547 1/20 0.41
CDC7 O00311 1/20 0.40
ROCK2 O75116 1/20 0.40
MAP4K4 O95819 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
PIM3 Q86V86 2/20 0.39
PIM2 Q9P1W9 2/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28911783 0.90 GSK3A (0.56) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28911710 0.89 GSK3B (0.51) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28911773 0.89 GSK3A (0.53) GSK3BGSK3AAURKBHDAC1
SCHEMBL20204977 0.85 GSK3B (0.67) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28911707 0.84 GSK3B (0.56) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28960743 0.84 GSK3A (0.51) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28911741 0.84 GSK3B (0.52) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28911743 0.83 GSK3A (0.61) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28911763 0.81 GSK3A (0.53) GSK3BGSK3APIM1CDK2JAK2
SCHEMBL28911730 0.81 GSK3A (0.49) GSK3BGSK3APIM1CDK2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110545817-B GSK-3 inhibitors 百时美施贵宝公司 2022-11-15 CN disclosed