SCHEMBL28925199

SCHEMBL28925199

COc1cc(N2CCC(N)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.59
MKNK1 Q9BUB5 1/20 0.57
MKNK2 Q9HBH9 1/20 0.57
HDAC1 Q13547 3/20 0.49
HDAC3 O15379 2/20 0.49
HDAC4 P56524 2/20 0.49
HDAC7 Q8WUI4 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC10 Q969S8 2/20 0.49
HDAC11 Q96DB2 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
HDAC9 Q9UKV0 2/20 0.49
HDAC5 Q9UQL6 2/20 0.49
JAK2 O60674 1/20 0.49
ROS1 P08922 1/20 0.49
PDGFRA P16234 1/20 0.49
FLT4 P35916 1/20 0.49
FLT3 P36888 1/20 0.49
MLNR O43193 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30070623 1.00 EGFR (0.59) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL29973838 0.92 EGFR (0.70) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL14663321 0.92 EGFR (0.70) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL28646094 0.92 EGFR (0.55) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL28639357 0.92 EGFR (0.55) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL28639358 0.92 EGFR (0.55) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL30070701 0.92 EGFR (0.55) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL19336981 0.91 EGFR (0.61) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL19337084 0.91 EGFR (0.63) EGFRMKNK1MKNK2HDAC1HDAC3
SCHEMBL19337010 0.91 EGFR (0.63) EGFRMKNK1MKNK2HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354622-B P-phenylenediamine LSD1 inhibitor and preparation method thereof 沈阳药科大学 2022-11-01 CN disclosed
CN-113354622-A P-phenylenediamine LSD1 inhibitor and preparation method thereof 沈阳药科大学 2021-09-07 CN disclosed