SCHEMBL28940950

SCHEMBL28940950

NC(=O)Oc1ccnc(OCCO)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
CHEK1 O14757 1/20 0.36
IKBKB O14920 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
CHEK2 O96017 1/20 0.34
ABL1 P00519 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RECQL P46063 1/20 0.34
KIF11 P52732 1/20 0.34
GAA P10253 1/20 0.34
LOXL2 Q9Y4K0 2/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CA1 P00915 2/20 0.32
MAOA P21397 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
LTB4R Q15722 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9572453 0.83 MEN1 (0.53) KMT2AMEN1ALDH1A1KIF11LOXL2
SCHEMBL28940925 0.81 CYP2D6 (0.46) KMT2AMEN1KIF11LOXL2HDAC1
SCHEMBL15881349 0.79 MEN1 (0.48) KMT2AMEN1LOXL2
SCHEMBL28941077 0.78 MEN1 (0.41) KMT2AMEN1KIF11LOXL2
SCHEMBL28941045 0.78 MEN1 (0.41) KMT2AMEN1LOXL2GCK
SCHEMBL28575456 0.78 CHEK2 (0.44) CHEK1IKBKBCHEK2HDAC1HDAC6
SCHEMBL28940998 0.77 MEN1 (0.40) KMT2AMEN1ABL1GCK
SCHEMBL28723920 0.76 GCK (0.40) KMT2AMEN1CHEK2ABL1ALDH1A1
SCHEMBL28292605 0.76 MEN1 (0.46) KMT2AMEN1ALDH1A1KIF11
SCHEMBL28292630 0.76 MEN1 (0.48) KMT2AMEN1ALDH1A1KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed