SCHEMBL28945558

SCHEMBL28945558

NCc1ccccc1-n1ncc(-c2ccc3nccnc3c2)c1Nc1ccccc1C(=O)O

nearest known ligand 0.76

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 12/20 0.76
ADORA2B P29275 2/20 0.51
ADORA3 P0DMS8 1/20 0.44
ADORA2A P29274 1/20 0.42
TGFBR1 P36897 1/20 0.37
FABP3 P05413 1/20 0.37
FABP4 P15090 1/20 0.37
FABP5 Q01469 1/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
FTO Q9C0B1 1/20 0.35
ROCK2 O75116 1/20 0.34
CLCN2 P51788 1/20 0.34
MAPK8 P45983 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27826568 0.91 ADORA1 (0.65) ADORA1ADORA2BADORA3ADORA2ATGFBR1
SCHEMBL3306156 0.86 ADORA1 (1.00) ADORA1ADORA2BADORA3ADORA2ATGFBR1
SCHEMBL3304067 0.85 ADORA1 (0.77) ADORA1ADORA2BADORA3ADORA2ATGFBR1
SCHEMBL1817011 0.78 ADORA1 (0.83) ADORA1ADORA2BADORA3ADORA2AKDM4E
SCHEMBL1817013 0.76 ADORA1 (0.81) ADORA1ADORA2BADORA3ADORA2ATGFBR1
SCHEMBL28790507 0.76 ADORA1 (0.42) ADORA1TGFBR1ALDH1A1GAAMAPT
SCHEMBL1816888 0.76 ADORA1 (0.67) ADORA1ADORA2BADORA3ADORA2ATGFBR1
SCHEMBL1816776 0.72 ADORA1 (0.68) ADORA1ADORA2BADORA3ADORA2ATGFBR1
SCHEMBL3305031 0.70 ADORA1 (1.00) ADORA1ADORA2BADORA3ADORA2A
SCHEMBL27637060 0.69 GRM5 (0.42) ADORA1KDM4EPOLBGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102197031-A Substituted 5-aminopyrazoles and use thereof BAYER SCHERING PHARMA AG 2011-09-21 CN disclosed