SCHEMBL28945950

SCHEMBL28945950

[2H]C([2H])([2H])c1nc(C(=O)OC)co1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 1/20 0.40
NPSR1 Q6W5P4 1/20 0.38
MAPK1 P28482 2/20 0.36
MAPT P10636 3/20 0.36
CYP1A2 P05177 2/20 0.36
TP53 P04637 2/20 0.36
GAA P10253 1/20 0.36
RECQL P46063 1/20 0.36
NPC1 O15118 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286492 0.87 DAGLA (0.43) DAGLANPSR1MAPK1MAPTCYP1A2
SCHEMBL161081 0.76 DAGLA (0.43) DAGLANPSR1MAPK1MAPTCYP1A2
SCHEMBL4484701 0.74 DAGLA (0.42) DAGLANPSR1MAPK1MAPTCYP1A2
SCHEMBL1027752 0.74 DAGLA (0.42) DAGLANPSR1MAPK1MAPTCYP1A2
SCHEMBL11921730 0.74 NPSR1 (0.40) NPSR1MAPK1MAPTCYP1A2TP53
SCHEMBL25234479 0.74 DAGLA (0.42) DAGLANPSR1MAPK1MAPTCYP1A2
SCHEMBL1196102 0.74 DAGLA (0.42) DAGLANPSR1MAPK1MAPTCYP1A2
SCHEMBL7324378 0.71 DAGLA (0.40) DAGLANPSR1MAPK1MAPTTP53
SCHEMBL16130104 0.71 DAGLA (0.43) DAGLANPSR1MAPK1
SCHEMBL77505 0.71 DAGLA (0.40) DAGLANPSR1MAPK1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115667273-A Competitive and non-competitive inhibitors of muscarinic acetylcholine receptor M5 范德堡大学 2023-01-31 CN disclosed