SCHEMBL28948680

SCHEMBL28948680

CC1CN(C(=O)c2ccc(F)c(F)c2)C=C(C(=O)O)c2[nH]c3ccccc3c21.NC(=O)C1CCC1

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 13/20 0.66
ESR1 P03372 2/20 0.44
NR3C1 P04150 1/20 0.44
PGR P06401 1/20 0.44
NR3C2 P08235 1/20 0.44
AR P10275 1/20 0.44
ABCB1 P08183 2/20 0.37
ABCG2 Q9UNQ0 2/20 0.37
SSTR3 P32745 2/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
MAPKAPK2 P49137 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6531590 0.93 NR1H4 (0.69) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL29880943 0.91 NR1H4 (0.77) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL689187 0.91 NR1H4 (0.77) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL272855 0.83 NR1H4 (0.68) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL688528 0.81 NR1H4 (0.76) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL6531592 0.81 NR1H4 (0.72) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL28819542 0.81 NR1H4 (0.43) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL4298714 0.80 NR1H4 (0.66) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL28948679 0.80 NR1H4 (0.70) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL274595 0.80 NR1H4 (1.00) NR1H4ESR1NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110404073-B Methods and pharmaceutical compositions for treating hepatitis B virus infection 国家医疗保健研究所 2022-08-16 CN disclosed