SCHEMBL28953154

SCHEMBL28953154

Cc1ccc(C(=O)N2Cc3[nH]nc(NC(=O)c4ccc(C(=O)O)cc4)c3C2)cc1

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AURKA O14965 18/20 0.76
CCNA2 P20248 9/20 0.76
CDK2 P24941 9/20 0.76
CCNA1 P78396 9/20 0.76
AURKB Q96GD4 4/20 0.50
ALK Q9UM73 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28841889 0.91 AURKA (0.76) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL28841828 0.90 AURKA (0.74) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL28841859 0.88 AURKA (0.71) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL28841876 0.87 CCNA2 (0.59) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL28953143 0.86 AURKA (0.69) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL2918134 0.86 AURKA (1.00) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL2922424 0.85 AURKA (0.80) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL28841936 0.83 AURKA (0.64) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL2916467 0.83 AURKA (0.72) AURKACCNA2CDK2CCNA1AURKB
SCHEMBL2922578 0.83 AURKA (0.75) AURKACCNA2CDK2CCNA1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115057860-B ERK inhibitor and pharmaceutical application thereof 四川大学华西医院 2024-02-09 CN disclosed
CN-115057860-A ERK inhibitor and pharmaceutical application thereof 四川大学华西医院 2022-09-16 CN disclosed