SCHEMBL28965181

SCHEMBL28965181

Nc1nc(N)c2c(-c3ccc(F)cc3)[nH]nc2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 8/20 0.48
PIK3CA P42336 8/20 0.48
PIK3CB P42338 8/20 0.48
PIK3CG P48736 8/20 0.48
PRKDC P78527 8/20 0.48
MAPK14 Q16539 2/20 0.47
ABL1 P00519 3/20 0.46
SRC P12931 2/20 0.46
MKNK1 Q9BUB5 3/20 0.44
MKNK2 Q9HBH9 1/20 0.44
ALK Q9UM73 2/20 0.43
GRM5 P41594 2/20 0.41
MAPT P10636 1/20 0.41
NUDT14 O95848 1/20 0.41
NUDT5 Q9UKK9 1/20 0.41
DAPK3 O43293 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
PAK4 O96013 1/20 0.40
NTRK1 P04629 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28960379 0.84 PIK3CD (0.64) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL28965180 0.84 PIK3CG (0.62) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL28960377 0.74 PIK3CD (0.67) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL28960378 0.71 PIK3CG (0.56) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL3424170 0.70 ABL1 (0.41) ABL1SRCEGFRPRKCA
SCHEMBL18040265 0.70 PIK3CD (0.60) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL2910349 0.70 ADORA2A (0.54) ABL1SRCMAPTEGFRPRKCA
SCHEMBL21711385 0.68 IKBKB (0.58) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20075417 0.68 MAPK1 (0.69) MAPK14ABL1SRCALKMAPT
SCHEMBL3417904 0.65 ABL1 (0.40) ABL1SRCMAPTGSK3BEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108371662-B Application of five-membered heterocyclic pyrimidine compound 中国药科大学 2023-03-03 CN claimed