SCHEMBL28972005

SCHEMBL28972005

COc1ccc2c(-c3ccc(OC(=O)C(=O)Oc4ccc(-c5ccnc6cc(OC)ccc56)cc4C)c(C)c3)ccnc2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 5/20 0.69
ENPP3 O14638 1/20 0.49
ENPP1 P22413 1/20 0.49
GRM4 Q14833 3/20 0.46
KCNH2 Q12809 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.42
HTR1A P08908 2/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
LMNA P02545 1/20 0.41
AURKA O14965 1/20 0.41
MET P08581 1/20 0.41
KDR P35968 1/20 0.41
TEK Q02763 1/20 0.41
AURKB Q96GD4 1/20 0.41
KDM5A P29375 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
KDM4E B2RXH2 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28972038 0.90 TLR8 (0.67) TLR8ENPP3ENPP1GRM4KCNH2
SCHEMBL28754511 0.90 TLR8 (0.67) TLR8ENPP3ENPP1GRM4KCNH2
SCHEMBL26420666 0.88 TLR8 (0.74) TLR8ENPP3ENPP1GRM4KCNH2
SCHEMBL31021032 0.85 TLR8 (0.67) TLR8ENPP3ENPP1GRM4KCNH2
SCHEMBL26128366 0.84 TLR8 (0.66) TLR8ENPP3ENPP1GRM4KCNH2
SCHEMBL26127884 0.84 TLR8 (0.65) TLR8ENPP3ENPP1GRM4KCNH2
SCHEMBL23496982 0.82 TLR8 (1.00) TLR8ENPP3ENPP1GRM4KCNH2
Oxalic Acid SCHEMBL28972006 0.81 TLR8 (0.88) TLR8ENPP3ENPP1GRM4KCNH2
Hydrochloric Acid SCHEMBL28754494 0.81 TLR8 (0.97) TLR8ENPP3ENPP1GRM4KCNH2
Hydrochloric Acid SCHEMBL29642045 0.81 TLR8 (0.97) TLR8ENPP3ENPP1GRM4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114702442-A 4- (7-methoxyquinoline-4-yl) -2-methylphenol malonate and preparation method thereof 北京拓领博泰生物科技有限公司 2022-07-05 CN disclosed