SCHEMBL28984084

SCHEMBL28984084

CC(=O)c1c(N)ncnc1NC(C)c1c(Cl)c2cccc(Cl)c2c(=O)n1-c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 12/20 0.61
PIK3R1 P27986 9/20 0.61
PIK3CG P48736 9/20 0.51
PIK3CB P42338 7/20 0.51
PIK3CA P42336 2/20 0.51
PIK3R2 O00459 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26246729 1.00 PIK3CD (0.61) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL30398158 1.00 PIK3CD (0.61) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL25396153 0.91 PIK3CD (0.52) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL30396632 0.91 PIK3CD (0.52) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL25396151 0.91 PIK3CD (0.52) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL26246743 0.86 PIK3CD (0.48) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL30426165 0.86 PIK3CD (0.48) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL26246747 0.86 PIK3CD (0.48) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
SCHEMBL26246712 0.83 PIK3CD (0.51) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA
Bosmolisib SCHEMBL20061373 0.80 PIK3CD (0.49) PIK3CDPIK3R1PIK3CGPIK3CBPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115968369-A Process for the preparation of compounds as PI3K inhibitors and intermediate compounds useful for the preparation thereof 株式会社保宁 2023-04-14 CN disclosed