SCHEMBL289902

SCHEMBL289902

COCCn1c(=O)sc2ccc(-c3ccc(CC(C#N)NC(=O)C4CCOCC4)cc3)cc21

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.72
KCNH2 Q12809 2/20 0.57
CTSK P43235 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2888750 0.85 CTSC (0.65) CTSCKCNH2CTSK
SCHEMBL2888743 0.85 CTSC (0.65) CTSCKCNH2CTSK
SCHEMBL288984 0.85 CTSC (0.72) CTSCKCNH2
SCHEMBL1499210 0.85 CTSC (0.72) CTSCKCNH2CTSK
SCHEMBL2072745 0.85 CTSC (0.72) CTSCKCNH2CTSK
SCHEMBL29433607 0.84 CTSC (1.00) CTSCKCNH2
SCHEMBL16932303 0.84 CTSC (1.00) CTSCKCNH2
SCHEMBL26117461 0.84 CTSC (1.00) CTSCKCNH2
SCHEMBL2892493 0.84 CTSC (0.63) CTSCKCNH2CTSK
Trifluoroacetic Acid SCHEMBL2890535 0.82 CTSC (0.61) CTSCKCNH2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP claimed
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed