SCHEMBL28995644

SCHEMBL28995644

CC(C)(C)OC(=O)NC(COCc1ccccc1)COc1ncc(Br)cc1Br

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.50
CTSS P25774 2/20 0.48
PPARG P37231 1/20 0.46
KLK7 P49862 2/20 0.43
KLK5 Q9Y337 2/20 0.43
SYK P43405 1/20 0.43
ATM Q13315 1/20 0.43
AAK1 Q2M2I8 6/20 0.43
RAB9A P51151 1/20 0.41
UGCG Q16739 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
CTSB P07858 1/20 0.39
CTSK P43235 1/20 0.39
CYP3A4 P08684 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30491809 1.00 PPARA (0.50) PPARACTSSPPARGKLK7KLK5
SCHEMBL25807391 1.00 PPARA (0.50) PPARACTSSPPARGKLK7KLK5
SCHEMBL30491806 0.91 PPARA (0.48) PPARACTSSPPARGKLK7KLK5
SCHEMBL28995593 0.91 PPARA (0.48) PPARACTSSPPARGKLK7KLK5
SCHEMBL25807459 0.91 PPARA (0.48) PPARACTSSPPARGKLK7KLK5
SCHEMBL28995695 0.89 ATM (0.53) CTSSKLK5ATMAAK1CTSB
SCHEMBL25811463 0.89 ATM (0.53) CTSSKLK5ATMAAK1CTSB
SCHEMBL25291935 0.87 UGCG (0.42) UGCG
SCHEMBL25252573 0.87 UGCG (0.42) UGCG
SCHEMBL30491783 0.86 PPARA (0.49) PPARACTSSPPARGKLK7KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916790-A Pyrido [2,3-b ] [1,4] oxazines or tetrahydropyrido [2,3-b ] [1,4] oxazepines as IAP antagonists 百济神州有限公司 2023-04-04 CN disclosed