SCHEMBL28995779

SCHEMBL28995779

NC(=O)OC(COCc1ccccc1)COc1ncc(Cl)cc1Br

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.39
UGCG Q16739 3/20 0.37
PSMB5 P28074 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC1A1 P43005 1/20 0.36
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
PPARA Q07869 1/20 0.35
TACR1 P25103 3/20 0.34
LNPEP Q9UIQ6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28995777 1.00 PLAU (0.39) PLAUUGCGPSMB5SLC6A4SLC1A1
SCHEMBL28995589 0.84 UGCG (0.40) UGCGPSMB5PPARA
SCHEMBL28995561 0.81 SLC1A1 (0.36) SLC1A1TACR1
SCHEMBL28995559 0.81 SLC1A1 (0.36) SLC1A1TACR1
SCHEMBL25296455 0.80 UGCG (0.41) PLAUUGCGPSMB5SLC6A4THRA
SCHEMBL25252120 0.80 UGCG (0.41) PLAUUGCGPSMB5SLC6A4THRA
SCHEMBL28995590 0.79 CYP1A2 (0.36)
SCHEMBL28995592 0.79 CYP1A2 (0.36)
SCHEMBL28995676 0.77 HDAC8 (0.38) PSMB5THRATHRBPPARA
SCHEMBL28995674 0.77 HDAC8 (0.38) PSMB5THRATHRBPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916790-A Pyrido [2,3-b ] [1,4] oxazines or tetrahydropyrido [2,3-b ] [1,4] oxazepines as IAP antagonists 百济神州有限公司 2023-04-04 CN disclosed