SCHEMBL28996166

SCHEMBL28996166

CS(=O)(=O)c1nccc(-c2cc(N)cc(-c3nccs3)n2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.47
SYK P43405 9/20 0.41
SRC P12931 5/20 0.41
ZAP70 P43403 4/20 0.41
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
CYP2C9 P11712 1/20 0.36
EDNRA P25101 1/20 0.36
SLC6A4 P31645 1/20 0.36
ADRA1A P35348 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CDK2 P24941 1/20 0.36
HPGD P15428 4/20 0.35
NPY5R Q15761 1/20 0.34
CRHR1 P34998 2/20 0.34
TLR7 Q9NYK1 1/20 0.34
EGFR P00533 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30252976 1.00 HSP90AA1 (0.47) HSP90AA1SYKSRCZAP70KDM4E
SCHEMBL24774090 0.87 DYRK1A (0.35) KDM4EALDH1A1LMNAHPGDEGFR
SCHEMBL29290793 0.84 HSP90AA1 (0.48) HSP90AA1SYKSRCZAP70CDK2
SCHEMBL30252756 0.80 ADORA2A (0.42) HSP90AA1SYKSRCZAP70KDM4E
SCHEMBL20911605 0.80 ADORA2A (0.42) HSP90AA1SYKSRCZAP70KDM4E
SCHEMBL30252762 0.80 HSP90AA1 (0.42) HSP90AA1SYKSRCZAP70CDK2
SCHEMBL20911603 0.80 HSP90AA1 (0.42) HSP90AA1SYKSRCZAP70CDK2
SCHEMBL30252529 0.78 HSP90AA1 (0.56) HSP90AA1SYKSRCZAP70ALDH1A1
SCHEMBL30252663 0.77 HSP90AA1 (0.49) HSP90AA1SYKSRCZAP70LMNA
SCHEMBL29290796 0.77 HSP90AA1 (0.42) HSP90AA1SYKSRCZAP70CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed