SCHEMBL28996972

SCHEMBL28996972

Cn1ncc2ccc(Nc3ncc(C(F)(F)F)c(Nc4ccccc4P(C)(C)=O)n3)cc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 3/20 0.54
EGFR P00533 7/20 0.52
KDR P35968 2/20 0.48
AURKB Q96GD4 1/20 0.48
PTK2 Q05397 4/20 0.47
CHEK1 O14757 1/20 0.46
FLT3 P36888 1/20 0.46
PTK2B Q14289 2/20 0.46
JAK2 O60674 1/20 0.46
NTRK1 P04629 1/20 0.46
TYK2 P29597 1/20 0.46
JAK3 P52333 1/20 0.46
NTRK3 Q16288 1/20 0.46
NTRK2 Q16620 1/20 0.46
CDC7 O00311 1/20 0.45
ROCK2 O75116 1/20 0.45
MAP4K4 O95819 1/20 0.45
PIM1 P11309 1/20 0.45
PRKACA P17612 1/20 0.45
CDK7 P50613 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28996874 0.86 EGFR (0.62) MAP4K1EGFRPTK2
SCHEMBL29833077 0.86 EGFR (0.62) MAP4K1EGFRPTK2
SCHEMBL30429476 0.84 PTK2 (0.48) KDRAURKBPTK2CHEK1FLT3
SCHEMBL29190521 0.84 PTK2 (0.56) EGFRKDRAURKBPTK2FLT3
SCHEMBL28996964 0.83 MAP4K1 (0.53) MAP4K1EGFRKDRAURKBPTK2
SCHEMBL30833740 0.82 PTK2 (0.50) KDRAURKBPTK2CHEK1FLT3
SCHEMBL30833667 0.82 KDR (0.48) KDRAURKBPTK2CHEK1FLT3
SCHEMBL30860863 0.81 LRRK2 (0.61) CHEK1FLT3JAK2ULK1
SCHEMBL27228258 0.81 LRRK2 (0.61) CHEK1FLT3JAK2ULK1
SCHEMBL31251206 0.80 EGFR (0.63) MAP4K1EGFRPTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116082399-A Condensed ring-2-aminopyrimidine compound, and composition and application thereof 浙江大学智能创新药物研究院 2023-05-09 CN disclosed