SCHEMBL28998232

SCHEMBL28998232

Cn1nnc(-c2cnc(NC(=O)C3(C#N)CC3)cn2)c1OC(N)=O

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.33
TBK1 Q9UHD2 2/20 0.31
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30352432 1.00 MKNK1 (0.33) MKNK1TBK1BTK
SCHEMBL28998194 0.87 AAK1 (0.35) MKNK1BTK
SCHEMBL28998255 0.83 BACE1 (0.33) MKNK1BTK
SCHEMBL28998213 0.82 BTK (0.35) BTK
SCHEMBL28998240 0.81 BACE1 (0.32) BTK
SCHEMBL28998733 0.79 BACE1 (0.39) BTK
SCHEMBL28998266 0.79
SCHEMBL28998149 0.78
SCHEMBL28998169 0.78 GSK3B (0.37)
SCHEMBL28998163 0.74 ATM (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115942972-A LPA receptor antagonists and uses thereof 吉利德科学公司 2023-04-07 CN disclosed