SCHEMBL2900919

SCHEMBL2900919

Brc1ccc2[nH]c(-c3n[nH]c4sccc34)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.44
ITK Q08881 14/20 0.43
CHEK1 O14757 1/20 0.40
CDK7 P50613 1/20 0.40
CLK2 P49760 2/20 0.38
DYRK1A Q13627 2/20 0.38
DCLK1 O15075 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
CHEK2 O96017 1/20 0.38
CSF1R P07333 1/20 0.38
FER P16591 1/20 0.38
CDK2 P24941 1/20 0.38
MARK3 P27448 1/20 0.38
FLT4 P35916 1/20 0.38
FLT3 P36888 1/20 0.38
MAPK9 P45984 1/20 0.38
CSNK1D P48730 1/20 0.38
CSNK2A1 P68400 1/20 0.38
CSNK1G2 P78368 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1622112 0.80 ITK (0.55) CYP19A1ITKCHEK1CDK7CLK2
SCHEMBL17422783 0.71 CYP19A1 (0.71) CYP19A1CHEK1FLT3CSNK2A1
SCHEMBL141689 0.69 ITK (0.73) ITKCHEK1CDK2
SCHEMBL15741187 0.67 MAPK1 (0.49) CHEK1CDK7CLK2DYRK1APRKD3
SCHEMBL17422896 0.66 CYP19A1 (0.59) CYP19A1CHEK1FLT3CSNK2A1
SCHEMBL17433444 0.65 CYP19A1 (0.62) CYP19A1ITKCHEK1DYRK1AFLT3
SCHEMBL6479098 0.64 CYP19A1 (0.53) CYP19A1ITKFLT3CSNK2A1
SCHEMBL15741280 0.64 TNKS2 (0.44) PDPK1
SCHEMBL17433446 0.64 CYP19A1 (0.61) CYP19A1ITKCHEK1FLT3CSNK2A1
SCHEMBL17422937 0.64 CYP19A1 (0.71) CYP19A1ITKCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682553-B1 THIENOPYRAZOLES AVENTIS PHARMA INC (US) 2010-05-19 EP disclosed