SCHEMBL29012252

SCHEMBL29012252

CC(=O)Nc1nnc(CC2CCSC2)c2cc(-c3ccc(Cl)cc3)sc12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 14/20 0.40
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MCHR1 Q99705 1/20 0.34
TP53 P04637 1/20 0.33
MDM2 Q00987 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MAP3K8 P41279 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29012210 0.95 CHEK1 (0.41) CHEK1MEN1NPC1LMNARAB9A
SCHEMBL29012207 0.85 CHEK1 (0.39) CHEK1MCHR1
SCHEMBL29012208 0.85 CHEK1 (0.49) CHEK1MCHR1
SCHEMBL29012233 0.84 CHEK1 (0.40) CHEK1MCHR1ALDH1A1KDM4E
SCHEMBL29012268 0.84 CHEK1 (0.53) CHEK1
SCHEMBL12921996 0.83 CHEK1 (0.42) CHEK1MEN1RAB9AKMT2ASMN1; SMN2
SCHEMBL8832476 0.82 CHEK1 (0.52) CHEK1MEN1RAB9AKMT2AALDH1A1
SCHEMBL8833455 0.81 CHEK1 (0.42) CHEK1MCHR1
SCHEMBL12922024 0.80 MAPT (0.39) CHEK1MEN1NPC1LMNARAB9A
SCHEMBL8831494 0.79 CHEK1 (0.42) CHEK1MEN1RAB9AKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115038439-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN claimed
CN-115038440-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN claimed
CN-115038439-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN disclosed
CN-115038440-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN disclosed