SCHEMBL2901422

SCHEMBL2901422

O=C1OC(c2ccc(Cl)cc2)CN1Cc1ccc(-c2cccc(CN3CCCCC3)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 6/20 0.52
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
FADS1 O60427 2/20 0.45
HRH3 Q9Y5N1 3/20 0.45
HTR2A P28223 1/20 0.44
LSS P48449 1/20 0.43
PRSS12 P56730 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LTA4H P09960 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HRH4 Q9H3N8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2892118 1.00 GRM2 (0.52) GRM2CYP2D6CYP2C19FADS1HRH3
SCHEMBL2892125 0.92 GRM2 (0.57) GRM2CYP2D6CYP2C19FADS1HRH3
SCHEMBL4329682 0.92 GRM2 (0.57) GRM2CYP2D6CYP2C19FADS1HRH3
SCHEMBL2893022 0.91 GRM2 (0.51) GRM2FADS1HRH3HTR2ALSS
SCHEMBL2893019 0.91 GRM2 (0.51) GRM2FADS1HRH3HTR2ALSS
SCHEMBL2896644 0.90 GRM2 (0.53) GRM2FADS1HTR2ALSSPRSS12
SCHEMBL13086193 0.90 GRM2 (0.50) GRM2CYP2C19FADS1HTR2ALSS
SCHEMBL2896643 0.90 GRM2 (0.53) GRM2FADS1HTR2ALSSPRSS12
SCHEMBL2901758 0.83 GRM2 (0.55) GRM2FADS1HTR2APRSS12
SCHEMBL2901760 0.83 GRM2 (0.55) GRM2FADS1HTR2APRSS12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070275966-A1 Oxazolidinone compounds and their use as metabotropic glutamate receptor potentiators NPS PHARMACEUTICALS, INC. (US) 2007-11-29 US claimed
US-7816354-B2 Oxazolidinone compounds and their use as metabotropic glutamate receptor potentiators ASTRAZENECA AB (SE) 2010-10-19 US disclosed
US-20090012089-A1 Oxazolidinone Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators ASTRAZENECA AB (SE) 2009-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275966-A1 Oxazolidinone compounds and their use as metabotropic glutamate receptor potentiators GRM1, GRIN1, GRM2 GRM2 3/4885CYP2D6 1230/4885CYP2C19 1244/4885
US-20090012089-A1 Oxazolidinone Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators GRM1, GRIN1, GRM2 GRM2 3/4885CYP2D6 1230/4885CYP2C19 1244/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.