SCHEMBL29020179

SCHEMBL29020179

CC(NC(=O)c1cc(-c2ccc(Cl)cc2)nc(-c2cnn(C)c2)n1)c1ccc(F)c(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 2/20 0.46
MAPK1 P28482 3/20 0.42
RET P07949 3/20 0.40
MET P08581 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
S1PR3 Q99500 3/20 0.39
S1PR4 O95977 1/20 0.38
S1PR1 P21453 1/20 0.38
EP300 Q09472 6/20 0.38
CSNK1D P48730 1/20 0.38
CSNK1E P49674 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29961651 1.00 CLK1 (0.46) CLK1MAPK1RETMETCNR1
SCHEMBL29020176 1.00 CLK1 (0.46) CLK1MAPK1RETMETCNR1
SCHEMBL29020204 0.94 CLK1 (0.46) CLK1MAPK1S1PR3S1PR4S1PR1
SCHEMBL29961565 0.94 CLK1 (0.46) CLK1MAPK1S1PR3S1PR4S1PR1
SCHEMBL29020202 0.94 CLK1 (0.46) CLK1MAPK1S1PR3S1PR4S1PR1
SCHEMBL29020159 0.90 CLK1 (0.50) CLK1MAPK1MET
SCHEMBL29961667 0.90 CLK1 (0.50) CLK1MAPK1MET
SCHEMBL29020156 0.90 CLK1 (0.50) CLK1MAPK1MET
SCHEMBL29020222 0.89 MAPK1 (0.52) CLK1MAPK1METCNR1
SCHEMBL29020226 0.89 MAPK1 (0.52) CLK1MAPK1METCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed