SCHEMBL29020194

SCHEMBL29020194

COc1ccc(-c2nc(C(=O)O)cc(-c3ccc(Cl)cc3)n2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.62
MCL1 Q07820 3/20 0.57
ADORA3 P0DMS8 6/20 0.53
PLA2G2A P14555 1/20 0.53
TP53 P04637 1/20 0.53
MAPT P10636 1/20 0.53
THRB P10828 1/20 0.53
KMO O15229 1/20 0.50
ADORA2B P29275 1/20 0.50
CHEK1 O14757 1/20 0.50
CTRC Q99895 1/20 0.49
HPGD P15428 1/20 0.49
PTPN1 P18031 1/20 0.48
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
AURKA O14965 1/20 0.48
AURKB Q96GD4 1/20 0.48
NPC1 O15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29962056 1.00 KDM4E (0.62) KDM4EMCL1ADORA3PLA2G2ATP53
SCHEMBL2928253 0.89 MCL1 (0.66) KDM4EMCL1ADORA3MAPTADORA2B
SCHEMBL21001267 0.89 MCL1 (0.61) KDM4EMCL1ADORA3KMOCTRC
SCHEMBL15383823 0.85 MCL1 (0.65) KDM4EMCL1PLA2G2ATP53MAPT
SCHEMBL29020197 0.82 MCL1 (0.55) KDM4EMCL1ADORA3MAPTKMO
SCHEMBL22391758 0.80 MAPT (0.47) KDM4EADORA3PLA2G2AMAPTADORA2B
SCHEMBL21004859 0.79 AHR (0.57) KDM4EADORA3PLA2G2ATP53MAPT
SCHEMBL21004858 0.79 AHR (0.57) KDM4EADORA3PLA2G2ATP53MAPT
SCHEMBL29020146 0.78 MCL1 (0.51) KDM4EMCL1ADORA3MAPTKMO
SCHEMBL29961510 0.78 MCL1 (0.51) KDM4EMCL1ADORA3MAPTKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed