SCHEMBL29023074

SCHEMBL29023074

COC(=O)c1cc(Br)c2cn[nH]c2c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
HPGD P15428 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
POLB P06746 4/20 0.37
NR4A2 P43354 2/20 0.37
METAP2 P50579 1/20 0.36
HSD17B10 Q99714 2/20 0.36
SOS1 Q07889 1/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30052019 1.00 TSHR (0.45) TSHRKDM4EALDH1A1HPGDNPSR1
SCHEMBL27186379 0.87 TSHR (0.44) TSHRKDM4EALDH1A1HPGDNPSR1
SCHEMBL31211411 0.79 TSHR (0.47) TSHRKDM4EALDH1A1L3MBTL1POLB
SCHEMBL21458300 0.79 TSHR (0.47) TSHRKDM4EALDH1A1L3MBTL1POLB
SCHEMBL27186999 0.77 HSD17B10 (0.49) TSHRKDM4EALDH1A1HPGDMETAP2
SCHEMBL29023121 0.77 JAK3 (0.42) TSHRKDM4EALDH1A1HPGDNPSR1
SCHEMBL30969311 0.77 TSHR (0.47) TSHRKDM4EALDH1A1L3MBTL1POLB
SCHEMBL31638752 0.76 TSHR (0.38) TSHRKDM4EALDH1A1HPGDNPSR1
SCHEMBL20577534 0.76 AXL (0.37) KDM4EALDH1A1HPGDMETAP2AXL
SCHEMBL12869690 0.75 PIM3 (0.47) KDM4EALDH1A1HPGDNPSR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116348453-A Heteroaromatic carboxamide compounds and uses thereof 烨辉医药科技(上海)有限公司 2023-06-27 CN disclosed
WO-2022228302-A1 HETEROAROMATIC CARBOXAMIDE COMPOUNDS AND ITS USE BIONOVA PHARMACEUTICALS (SHANGHAI) LIMITED (CN) 2022-11-03 WO disclosed