SCHEMBL29036015

SCHEMBL29036015

CC(C)(C)OC(=O)NC1(C(=O)NC(C(=O)O)c2ccccc2)CCN(c2ncnc3[nH]ccc23)CC1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 15/20 0.58
ROCK2 O75116 10/20 0.57
AKT2 P31751 10/20 0.57
AKT3 Q9Y243 10/20 0.57
KCNH2 Q12809 6/20 0.52
JAK3 P52333 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29036005 1.00 AKT1 (0.58) AKT1ROCK2AKT2AKT3KCNH2
SCHEMBL29157947 0.94 AKT1 (0.57) AKT1ROCK2AKT2AKT3KCNH2
SCHEMBL30012817 0.94 AKT1 (0.57) AKT1ROCK2AKT2AKT3KCNH2
SCHEMBL29157946 0.94 AKT1 (0.57) AKT1ROCK2AKT2AKT3KCNH2
SCHEMBL390393 0.88 AKT1 (0.70) AKT1ROCK2AKT2AKT3KCNH2
SCHEMBL390394 0.88 AKT1 (0.70) AKT1ROCK2AKT2AKT3KCNH2
SCHEMBL31374403 0.84 JAK3 (0.58) AKT1ROCK2AKT2AKT3JAK3
SCHEMBL390884 0.84 JAK3 (0.58) AKT1ROCK2AKT2AKT3JAK3
SCHEMBL391355 0.82 AKT1 (0.71) AKT1ROCK2AKT2AKT3KCNH2
SCHEMBL10156733 0.82 AKT1 (0.64) AKT1ROCK2AKT2AKT3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232130-A APN and AKT double-target-point inhibitor and preparation method and application thereof 山东大学 2022-10-25 CN disclosed