SCHEMBL2904232

SCHEMBL2904232

COc1cc2ncc(C(N)=O)c(Nc3cccc(Cl)c3F)c2cc1N1CCN(C)CC1

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 17/20 0.79
KCNH2 Q12809 4/20 0.72
SCN5A Q14524 3/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912082 0.97 CSF1R (0.85) CSF1RKCNH2SCN5A
SCHEMBL1276321 0.92 KCNH2 (0.85) CSF1RKCNH2SCN5A
SCHEMBL2912771 0.92 CSF1R (0.93) CSF1RKCNH2SCN5A
SCHEMBL2905870 0.91 KCNH2 (0.72) CSF1RKCNH2SCN5A
SCHEMBL2912060 0.91 KCNH2 (0.69) CSF1RKCNH2SCN5A
SCHEMBL2908557 0.91 CSF1R (0.80) CSF1RKCNH2SCN5A
SCHEMBL2907805 0.91 KCNH2 (0.73) CSF1RKCNH2SCN5A
SCHEMBL2908767 0.89 CSF1R (0.83) CSF1RKCNH2SCN5A
SCHEMBL2912249 0.89 KCNH2 (0.64) CSF1RKCNH2SCN5A
SCHEMBL2913716 0.89 CSF1R (0.88) CSF1RKCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed