SCHEMBL2904510

SCHEMBL2904510

CCOC(=O)c1cnc2cc(OC)c(N3CCN(CC)CC3)cc2c1Nc1cccc(Cl)c1Cl

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.65
SCN5A Q14524 1/20 0.65
CSF1R P07333 13/20 0.64
MAPT P10636 2/20 0.53
GAA P10253 1/20 0.53
THRB P10828 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904857 0.97 KCNH2 (0.61) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2908314 0.97 CSF1R (0.69) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2909867 0.94 KCNH2 (0.72) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2907631 0.93 KCNH2 (0.75) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2910713 0.92 KCNH2 (0.68) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2913141 0.91 KCNH2 (0.68) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2914058 0.91 KCNH2 (0.63) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2907259 0.91 KCNH2 (0.65) KCNH2SCN5ACSF1RMAPTGAA
SCHEMBL2913800 0.91 CSF1R (0.78) KCNH2SCN5ACSF1R
SCHEMBL2911776 0.90 KCNH2 (0.71) KCNH2SCN5ACSF1RMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed