SCHEMBL2904843

SCHEMBL2904843

CCOC(=O)c1cnc2cc(F)c(N3CCOCC3)cc2c1Nc1ccc(F)cc1F

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 6/20 0.63
KCNH2 Q12809 6/20 0.61
SCN5A Q14524 2/20 0.61
MAPT P10636 7/20 0.56
GAA P10253 6/20 0.56
LMNA P02545 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
MC4R P32245 2/20 0.56
HTT P42858 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
PTK2B Q14289 1/20 0.56
MAPK1 P28482 1/20 0.55
CLK1 P49759 1/20 0.55
GSK3A P49840 1/20 0.55
GSK3B P49841 1/20 0.55
TP53 P04637 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912345 0.94 CSF1R (0.71) CSF1RKCNH2SCN5AMAPTGAA
SCHEMBL2904374 0.92 CSF1R (0.66) CSF1RKCNH2SCN5AMAPTGAA
SCHEMBL2904098 0.91 CSF1R (0.77) CSF1RKCNH2SCN5AGAAMEN1
SCHEMBL2913762 0.88 MAPT (0.68) CSF1RKCNH2SCN5AMAPTGAA
SCHEMBL2908692 0.86 CSF1R (0.80) CSF1RKCNH2SCN5A
SCHEMBL2911029 0.85 CSF1R (0.84) CSF1RKCNH2SCN5AGAAMEN1
SCHEMBL2911267 0.85 CSF1R (0.72) CSF1RKCNH2SCN5A
SCHEMBL2913291 0.84 CSF1R (0.85) CSF1RKCNH2SCN5A
SCHEMBL2910570 0.84 KCNH2 (0.84) CSF1RKCNH2SCN5AMAPTLMNA
SCHEMBL2909944 0.84 CSF1R (0.78) CSF1RKCNH2SCN5AGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed