SCHEMBL2905342

SCHEMBL2905342

CCOC(=O)c1cnc2cc(OCC)c(N3CCCN(C)CC3)cc2c1Nc1ccc(F)cc1F

nearest known ligand 0.84

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.84
CSF1R P07333 10/20 0.79
SCN5A Q14524 5/20 0.79
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
GAA P10253 1/20 0.48
SLC2A1 P11166 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2911029 0.97 CSF1R (0.84) KCNH2CSF1RSCN5AMEN1KMT2A
SCHEMBL2911256 0.95 KCNH2 (0.76) KCNH2CSF1RSCN5AMEN1KMT2A
SCHEMBL2912797 0.94 KCNH2 (0.75) KCNH2CSF1RSCN5AMEN1KMT2A
SCHEMBL2909944 0.94 CSF1R (0.78) KCNH2CSF1RSCN5AMEN1KMT2A
SCHEMBL2912694 0.92 KCNH2 (0.71) KCNH2CSF1RSCN5A
SCHEMBL2913031 0.92 CSF1R (0.75) KCNH2CSF1RSCN5AMEN1KMT2A
SCHEMBL2910877 0.92 KCNH2 (1.00) KCNH2CSF1RSCN5A
SCHEMBL2904648 0.92 CSF1R (0.79) KCNH2CSF1RSCN5AMEN1KMT2A
SCHEMBL2905716 0.91 CSF1R (0.73) KCNH2CSF1RSCN5AMEN1KMT2A
SCHEMBL2910730 0.91 KCNH2 (0.85) KCNH2CSF1RSCN5AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed