SCHEMBL29064455

SCHEMBL29064455

Nc1ncnc2c1c(I)cn2C[C@H]1CCCN1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 17/20 0.47
DYRK3 O43781 1/20 0.46
ROCK2 O75116 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
PHKG2 P15735 1/20 0.46
PRKACA P17612 1/20 0.46
RPS6KB1 P23443 1/20 0.46
MARK3 P27448 1/20 0.46
FLT3 P36888 1/20 0.46
CSNK1A1 P48729 1/20 0.46
CSNK1D P48730 1/20 0.46
CLK2 P49760 1/20 0.46
IRAK1 P51617 1/20 0.46
CSNK1G2 P78368 1/20 0.46
MAP4K2 Q12851 1/20 0.46
ROCK1 Q13464 1/20 0.46
CAMK2G Q13555 1/20 0.46
CAMK2D Q13557 1/20 0.46
DYRK1A Q13627 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15564132 1.00 BTK (0.47) BTKDYRK3ROCK2PRKD3MAP4K4
SCHEMBL28097476 1.00 BTK (0.47) BTKDYRK3ROCK2PRKD3MAP4K4
SCHEMBL29064399 0.87 BTK (0.39) BTKFGFR1FGFR4LCKFYN
SCHEMBL29064397 0.87 BTK (0.39) BTKFGFR1FGFR4LCKFYN
SCHEMBL13858252 0.85 BTK (0.47) BTKFGFR1FGFR4SRC
SCHEMBL13858254 0.85 BTK (0.47) BTKFGFR1FGFR4SRC
SCHEMBL16769872 0.85 BTK (0.47) BTKFGFR1FGFR4SRC
SCHEMBL20981724 0.81 FLT3 (0.42) BTKDYRK3ROCK2PRKD3MAP4K4
SCHEMBL15515675 0.80 BTK (0.53) BTKDYRK3PRKD3MAP4K4PRKACA
SCHEMBL13860235 0.80 BTK (0.53) BTKDYRK3PRKD3MAP4K4PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514806-A Biological inhibitor containing acrylketone, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-08-01 CN disclosed