SCHEMBL2906861

SCHEMBL2906861

COc1ccc(CNc2ccc3ncc(C(=O)Nc4ccc(C(=O)O)cc4)n3n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FYN P06241 8/20 0.51
PIM1 P11309 2/20 0.48
HDAC1 Q13547 1/20 0.46
P4HTM Q9NXG6 1/20 0.45
NTRK1 P04629 1/20 0.44
CLK1 P49759 2/20 0.44
VNN1 O95497 1/20 0.43
HIF1A Q16665 1/20 0.43
ALDH1A1 P00352 1/20 0.43
IKBKB O14920 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1203239 0.91 FYN (0.51) FYNPIM1HDAC1NTRK1CLK1
SCHEMBL1203328 0.91 FYN (0.55) FYNPIM1HDAC1NTRK1CLK1
SCHEMBL1203735 0.91 FYN (0.52) FYNPIM1HDAC1NTRK1CLK1
SCHEMBL1203488 0.90 FYN (0.52) FYNPIM1NTRK1CLK1ALDH1A1
SCHEMBL1203065 0.89 PPARA (0.54) FYNPIM1HDAC1NTRK1
SCHEMBL1202563 0.89 MEN1 (0.53) FYNPIM1HDAC1NTRK1ALDH1A1
SCHEMBL1202181 0.87 FYN (0.49) FYNPIM1HDAC1NTRK1VNN1
SCHEMBL1203600 0.86 FYN (0.59) FYNPIM1NTRK1CLK1VNN1
SCHEMBL1202889 0.86 PIM1 (0.50) FYNPIM1HDAC1NTRK1VNN1
SCHEMBL2943172 0.84 FYN (0.69) FYNPIM1NTRK1IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217601-A1 IMIDAZOPYRIDAZINES FOR USE AS PROTEIN KINASE INHIBITORS Centro Nacional de Investigaciones Oncológicas (CNIO) (ES) 2010-08-18 EP disclosed
WO-2009060197-A1 IMIDAZOPYRIDAZINES FOR USE AS PROTEIN KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2009-05-14 WO disclosed