SCHEMBL2907438

SCHEMBL2907438

NC(=O)c1noc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 18/20 0.58
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
LMNA P02545 1/20 0.46
CA3 P07451 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
MAOB P27338 1/20 0.46
CA5A P35218 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA13 Q8N1Q1 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
LCK P06239 1/20 0.43
MAP2K3 P46734 1/20 0.43
MAP2K6 P52564 1/20 0.43
BTK Q06187 1/20 0.43
MAP3K19 Q56UN5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29580724 1.00 HIF1A (0.58) HIF1ACA12CA1CA2LMNA
Cyclohexane SCHEMBL2442670 0.95 HIF1A (0.58) HIF1ACA12CA1CA2LMNA
SCHEMBL2448188 0.85 HIF1A (0.46) HIF1A
Benzothiophene SCHEMBL2439236 0.83 HIF1A (0.44) HIF1A
SCHEMBL496601 0.82 HIF1A (0.65) HIF1A
SCHEMBL9046980 0.82 HIF1A (0.43) HIF1A
SCHEMBL1809709 0.81 HIF1A (0.58) HIF1A
SCHEMBL3434886 0.81 HIF1A (0.61) HIF1A
SCHEMBL20189383 0.80 HIF1A (0.67) HIF1A
SCHEMBL29581929 0.80 HIF1A (0.56) HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115677608-B Benzisoxazole-3-carboxamide compound and synthesis and application thereof 复旦大学 2024-06-07 CN claimed
CN-117836306-A Galactose glycoside derivatives as galectin-3 inhibitors 株式会社蒂奥姆生物 2024-04-05 CN claimed
EP-3472149-B1 HETEROCYCLIC PROLINAMIDE DERIVATIVES Orion Ophthalmology LLC (US) 2023-08-30 EP claimed
CN-115677608-A Benzisoxazole-3-formamide compound and synthesis and application thereof 复旦大学 2023-02-03 CN claimed
US-12281101-B2 Bicyclic lactams and methods of use thereof GENENTECH, INC. (US) 2025-04-22 US disclosed
CN-115677608-B Benzisoxazole-3-carboxamide compound and synthesis and application thereof 复旦大学 2024-06-07 CN disclosed
CN-115677608-B Benzisoxazole-3-carboxamide compound and synthesis and application thereof 复旦大学 2024-06-07 CN disclosed
CN-115677608-B Benzisoxazole-3-carboxamide compound and synthesis and application thereof 复旦大学 2024-06-07 CN disclosed
CN-117836306-A Galactose glycoside derivatives as galectin-3 inhibitors 株式会社蒂奥姆生物 2024-04-05 CN disclosed
CN-115677608-A Benzisoxazole-3-formamide compound and synthesis and application thereof 复旦大学 2023-02-03 CN disclosed
CN-115677608-A Benzisoxazole-3-formamide compound and synthesis and application thereof 复旦大学 2023-02-03 CN disclosed
CN-115677608-A Benzisoxazole-3-formamide compound and synthesis and application thereof 复旦大学 2023-02-03 CN disclosed
US-5225412-A Antipsychotic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-06 US disclosed
US-5225412-A Antipsychotic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-06 US disclosed
EP-0511610-A1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-04 EP disclosed
EP-0511610-A1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-04 EP disclosed
EP-0511610-A1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-04 EP disclosed
US-5143923-A Psychological disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-09-01 US disclosed
US-5143923-A Psychological disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-09-01 US disclosed
US-5143923-A Psychological disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12281101-B2 Bicyclic lactams and methods of use thereof LSS, LPXN, CYP1B1 HIF1A 3643/4885CA12 2507/4885CA1 2491/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.