SCHEMBL29080511

SCHEMBL29080511

N#CCCC1CCC(n2cc(-c3ncnc4[nH]ccc34)cn2)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 19/20 0.53
JAK1 P23458 18/20 0.53
JAK3 P52333 9/20 0.53
TYK2 P29597 4/20 0.53
RET P07949 3/20 0.53
ROCK1 Q13464 3/20 0.53
DAPK3 O43293 2/20 0.53
PAK4 O96013 2/20 0.53
ABL1 P00519 2/20 0.53
LTK P29376 2/20 0.53
CSNK1A1 P48729 2/20 0.53
CLK2 P49760 2/20 0.53
TNK2 Q07912 2/20 0.53
DYRK1A Q13627 2/20 0.53
IKBKE Q14164 2/20 0.53
NTRK3 Q16288 2/20 0.53
NTRK2 Q16620 2/20 0.53
LRRK2 Q5S007 2/20 0.53
TAOK1 Q7L7X3 2/20 0.53
CAMK1D Q8IU85 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phosphoric Acid SCHEMBL27231611 0.95 JAK2 (0.57) JAK2JAK1JAK3TYK2RET
SCHEMBL101257 0.94 JAK2 (0.55) JAK2JAK1JAK3TYK2RET
SCHEMBL101258 0.94 JAK2 (0.55) JAK2JAK1JAK3TYK2RET
SCHEMBL13774673 0.94 JAK2 (0.55) JAK2JAK1JAK3TYK2RET
SCHEMBL30663312 0.87 JAK2 (0.57) JAK2JAK1JAK3TYK2RET
SCHEMBL101692 0.87 JAK2 (0.57) JAK2JAK1JAK3TYK2RET
SCHEMBL101693 0.87 JAK2 (0.57) JAK2JAK1JAK3TYK2RET
Trifluoroacetic Acid SCHEMBL99863 0.87 JAK2 (0.49) JAK2JAK1JAK3TYK2RET
SCHEMBL101170 0.86 JAK2 (0.56) JAK2JAK1JAK3TYK2RET
SCHEMBL99389 0.82 JAK2 (0.52) JAK2JAK1JAK3TYK2RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120055-A Combination therapy comprising a JAK pathway inhibitor and a ROCK inhibitor 因赛特公司 2023-11-24 CN claimed
CN-117964625-A Preparation method of high-optical-purity ponatinib intermediate 安徽万邦医药科技股份有限公司 2024-05-03 CN disclosed
CN-117120055-A Combination therapy comprising a JAK pathway inhibitor and a ROCK inhibitor 因赛特公司 2023-11-24 CN disclosed
CN-116879450-A Method for separating and purifying reed-keatinib precursor by using supercritical fluid chromatography system 江苏汉邦科技股份有限公司 2023-10-13 CN disclosed
CN-116761792-A Methods and intermediates for preparing JAK inhibitors 因赛特公司 2023-09-15 CN disclosed