SCHEMBL2908158

SCHEMBL2908158

CCOc1cc2ncc(C(N)=O)c(Nc3ccc(CC)cc3)c2cc1N1CCCN(C)CC1

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.72
CSF1R P07333 13/20 0.66
SCN5A Q14524 3/20 0.66
MEN1 O00255 1/20 0.49
GAA P10253 1/20 0.49
SLC2A1 P11166 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2914405 0.97 CSF1R (0.70) KCNH2CSF1RSCN5AMEN1GAA
SCHEMBL2911092 0.92 KCNH2 (0.61) KCNH2CSF1RSCN5AMEN1GAA
SCHEMBL2911569 0.89 CSF1R (0.60) KCNH2CSF1RSCN5A
SCHEMBL2910805 0.89 CSF1R (0.79) KCNH2CSF1RSCN5A
SCHEMBL2912323 0.88 CSF1R (0.59) KCNH2CSF1RSCN5AMEN1GAA
SCHEMBL2913282 0.88 GAA (0.62) KCNH2CSF1RSCN5AMEN1GAA
SCHEMBL2907474 0.88 KCNH2 (0.72) KCNH2CSF1RSCN5A
SCHEMBL2910987 0.87 KCNH2 (0.74) KCNH2CSF1RSCN5A
SCHEMBL2912644 0.86 KCNH2 (0.70) KCNH2CSF1RSCN5A
SCHEMBL2904662 0.85 CSF1R (0.84) KCNH2CSF1RSCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed