SCHEMBL2908233

SCHEMBL2908233

CCOc1cc2ncc(C(N)=O)c(Nc3cc(F)ccc3F)c2cc1N1CCCN(C)CC1

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.88
CSF1R P07333 14/20 0.83
SCN5A Q14524 3/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2907540 0.97 CSF1R (0.88) KCNH2CSF1RSCN5A
SCHEMBL2910877 0.94 KCNH2 (1.00) KCNH2CSF1RSCN5A
SCHEMBL2912493 0.93 KCNH2 (0.83) KCNH2CSF1RSCN5A
SCHEMBL2912797 0.92 KCNH2 (0.75) KCNH2CSF1RSCN5A
SCHEMBL29411758 0.91 CSF1R (1.00) KCNH2CSF1RSCN5A
SCHEMBL1276777 0.91 CSF1R (1.00) KCNH2CSF1RSCN5A
SCHEMBL2912237 0.91 CSF1R (0.77) KCNH2CSF1RSCN5A
SCHEMBL1276299 0.90 KCNH2 (0.88) KCNH2CSF1RSCN5A
SCHEMBL2912729 0.90 CSF1R (0.78) KCNH2CSF1RSCN5A
SCHEMBL2904081 0.89 CSF1R (0.87) KCNH2CSF1RSCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed