SCHEMBL2908263

SCHEMBL2908263

COc1c(/C=C/c2ccc(NS(C)(=O)=O)cc2)cc(-n2c(=O)[nH]cc(F)c2=O)cc1C(C)(C)C

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.57
CRBN Q96SW2 1/20 0.41
KIF11 P52732 1/20 0.32
TNFRSF1A P19438 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479100 0.86 CYP3A4 (0.61) CYP3A4CRBNTNFRSF1APTGS2
Water SCHEMBL2484221 0.85 CYP3A4 (0.60) CYP3A4CRBNTNFRSF1APTGS2
Water SCHEMBL2908232 0.84 CYP3A4 (0.59) CYP3A4CRBNTNFRSF1A
SCHEMBL2112795 0.82 CYP3A4 (0.56) CYP3A4CRBNTNFRSF1A
SCHEMBL2112792 0.82 CYP3A4 (0.56) CYP3A4CRBNTNFRSF1A
SCHEMBL1530185 0.82 CYP3A4 (0.56) CYP3A4CRBNKIF11
SCHEMBL1530182 0.82 CYP3A4 (0.56) CYP3A4CRBNKIF11
Abt-072 SCHEMBL479128 0.80 CRBN (0.63) CYP3A4CRBNTNFRSF1A
Abt-072 SCHEMBL1530682 0.80 CRBN (0.63) CYP3A4CRBNTNFRSF1A
Abt-072 SCHEMBL479219 0.80 CRBN (0.63) CYP3A4CRBNTNFRSF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222646-A1 URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C Abbott Laboratories (US) 2010-09-01 EP disclosed
EP-2203430-A1 N-PHENYL-DIOXO-HYDROPYRIMIDINES USEFUL AS HEPATITIS C VIRUS (HCV) INHIBITORS Abbott Laboratories (US) 2010-07-07 EP disclosed
WO-2009039127-A1 URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C ABBOTT LABORATORIES (US) 2009-03-26 WO disclosed
WO-2009039135-A1 N-PHENYL-DIOXO-HYDROPYRIMIDINES USEFUL AS HEPATITIS C VIRUS (HCV) INHIBITORS ABBOTT LABORATORIES (US) 2009-03-26 WO disclosed