SCHEMBL29089211

SCHEMBL29089211

c1ccc2oc(-n3cnc4cncnc43)nc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 3/20 0.42
GABRD O14764 3/20 0.42
GABRA1 P14867 3/20 0.42
GABRB1 P18505 3/20 0.42
GABRG2 P18507 3/20 0.42
GABRB3 P28472 3/20 0.42
GABRA5 P31644 3/20 0.42
GABRA3 P34903 3/20 0.42
GABRA2 P47869 3/20 0.42
GABRB2 P47870 3/20 0.42
GABRA4 P48169 3/20 0.42
GABRE P78334 3/20 0.42
GABRA6 Q16445 3/20 0.42
GABRG1 Q8N1C3 3/20 0.42
GABRG3 Q99928 3/20 0.42
GABRQ Q9UN88 3/20 0.42
CHRNA7 P36544 1/20 0.38
HTR3A P46098 1/20 0.38
EGFR P00533 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5984515 0.77 HTT (0.51) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL680855 0.73 FGFR1 (0.56) EGFRMKNK2CYP1A2TSHRCYP3A4
Hydrochloric Acid SCHEMBL4456679 0.72 FGFR1 (0.54) EGFRMKNK2CYP1A2TSHRCYP3A4
SCHEMBL26126509 0.70 BCHE (0.42) HTR3AMKNK2CYP1A2TSHRCYP3A4
SCHEMBL27754086 0.70 PDE10A (0.44) EGFRMKNK2CYP1A2TSHRCYP3A4
SCHEMBL30677290 0.70 CYP1A2 (0.46) GABRG2GABRB3GABRA5MKNK2CYP1A2
SCHEMBL4542537 0.70 POLB (0.54) MKNK2CYP1A2TSHRCYP3A4CLK4
SCHEMBL29240138 0.70 PI4KA (0.57) GABRG2GABRB3GABRA5EGFRMKNK2
SCHEMBL6944930 0.69 PI4KA (0.55) GABRG2GABRB3GABRA5MKNK2CYP1A2
SCHEMBL6942099 0.69 MKNK2 (0.40) GABRG2GABRB3GABRA5MKNK2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116903586-A Bicyclic heteroaryl containing compounds 正大天晴药业集团股份有限公司 2023-10-20 CN disclosed