SCHEMBL2909753

SCHEMBL2909753

Nc1nc(NCCCn2cc(C(=O)NCc3ccccc3)c(-c3ccc(Cl)cc3Cl)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
GSK3B P49841 4/20 0.46
GSK3A P49840 3/20 0.46
CDK1 P06493 2/20 0.44
POLB P06746 1/20 0.44
CCNB2 O95067 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNB3 Q8WWL7 1/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SIRT6 Q8N6T7 1/20 0.40
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CNR1 P21554 3/20 0.40
SIRT5 Q9NXA8 2/20 0.40
GAA P10253 1/20 0.37
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904255 0.93 GSK3B (0.47) HPGDCYP1A2CYP3A4CYP2C19GSK3B
SCHEMBL2903991 0.92 POLB (0.56) HPGDCYP1A2CYP3A4CYP2C19GSK3B
SCHEMBL2913492 0.91 GSK3B (0.45) HPGDCYP1A2CYP3A4CYP2C19GSK3B
SCHEMBL2904086 0.90 HPGD (0.45) HPGDCYP1A2CYP3A4GSK3BGSK3A
SCHEMBL2911606 0.89 GSK3B (0.48) HPGDCYP1A2CYP3A4CYP2C19GSK3B
SCHEMBL2909523 0.89 GSK3B (0.48) HPGDCYP2C19GSK3BGSK3ACDK1
SCHEMBL2910338 0.89 GSK3B (0.45) HPGDCYP1A2CYP3A4CYP2C19GSK3B
SCHEMBL2910223 0.89 GSK3B (0.48) CYP2C19GSK3BGSK3ACDK1POLB
SCHEMBL2904121 0.89 GSK3B (0.44) HPGDGSK3BGSK3ACDK1POLB
SCHEMBL1219415 0.88 GSK3B (0.51) GSK3BGSK3ACDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed