SCHEMBL2909768

SCHEMBL2909768

CCOC(=O)c1cnc2cc(OCCOC)c(N3CCN(C)CC3)cc2c1Nc1cc(C)ccc1F

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.65
SCN5A Q14524 6/20 0.65
CSF1R P07333 9/20 0.58
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
GAA P10253 2/20 0.49
SLC2A1 P11166 1/20 0.49
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
MC4R P32245 1/20 0.48
HTT P42858 1/20 0.48
PTK2B Q14289 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909206 0.94 CSF1R (0.64) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2910626 0.94 KCNH2 (0.74) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2907152 0.93 KCNH2 (0.75) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2907777 0.92 KCNH2 (0.67) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2912075 0.92 KCNH2 (0.61) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL1276327 0.91 KCNH2 (0.76) KCNH2SCN5ACSF1R
SCHEMBL2912359 0.91 CSF1R (0.63) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2913052 0.90 KCNH2 (0.71) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2904820 0.90 CSF1R (0.73) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2904655 0.88 CSF1R (0.59) KCNH2SCN5ACSF1RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed