SCHEMBL2910657

SCHEMBL2910657

CCOC(=O)c1cnc2cc(OC)c(N3CCN(C)CC3)cc2c1Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.79

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 12/20 0.79
GAA P10253 3/20 0.61
MEN1 O00255 1/20 0.61
SLC2A1 P11166 1/20 0.61
KMT2A Q03164 1/20 0.61
KCNH2 Q12809 3/20 0.56
SCN5A Q14524 3/20 0.56
BRD4 O60885 1/20 0.55
MAPT P10636 2/20 0.51
PAK1 Q13153 1/20 0.51
THRB P10828 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912636 0.97 CSF1R (0.75) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2908777 0.97 CSF1R (0.79) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2911202 0.94 CSF1R (0.70) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2913908 0.93 CSF1R (0.68) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2910769 0.93 CSF1R (0.68) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2907640 0.92 CSF1R (0.66) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2907416 0.91 CSF1R (0.66) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2905926 0.91 CSF1R (0.66) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2911379 0.91 CSF1R (0.66) CSF1RGAAMEN1SLC2A1KMT2A
SCHEMBL2911375 0.91 CSF1R (0.66) CSF1RGAAMEN1SLC2A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed