SCHEMBL29115463

SCHEMBL29115463

CC(O)CNC(=O)c1ccc(N2CCNCC2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.46
ALDH1A1 P00352 4/20 0.45
HPGD P15428 3/20 0.45
TSHR P16473 1/20 0.45
RAB9A P51151 3/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 3/20 0.44
MEN1 O00255 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
USP28 Q96RU2 3/20 0.43
USP25 Q9UHP3 2/20 0.43
GAA P10253 1/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NAMPT P43490 2/20 0.42
DDR1 Q08345 1/20 0.42
TLR2 O60603 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29961330 1.00 MAPT (0.46) MAPTALDH1A1HPGDTSHRRAB9A
SCHEMBL29115549 1.00 MAPT (0.46) MAPTALDH1A1HPGDTSHRRAB9A
SCHEMBL29960900 1.00 MAPT (0.46) MAPTALDH1A1HPGDTSHRRAB9A
SCHEMBL29115460 1.00 MAPT (0.46) MAPTALDH1A1HPGDTSHRRAB9A
SCHEMBL531966 0.85 MAPT (0.53) MAPTALDH1A1HPGDTSHRRAB9A
Hydrochloric Acid SCHEMBL708105 0.84 MAPT (0.52) MAPTALDH1A1HPGDTSHRRAB9A
SCHEMBL719372 0.83 MAPT (0.50) MAPTALDH1A1HPGDTSHRRAB9A
SCHEMBL29960627 0.82 MAPT (0.47) MAPTALDH1A1HPGDTSHRRAB9A
SCHEMBL29115582 0.82 MAPT (0.47) MAPTALDH1A1HPGDTSHRRAB9A
Hydrochloric Acid SCHEMBL710508 0.82 MAPT (0.49) MAPTALDH1A1HPGDTSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed