SCHEMBL2911892

SCHEMBL2911892

CCOC(=O)c1cnc2cc(OC)c(N3CCN(C)CC3)cc2c1Nc1ccc(C)cc1F

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.76
SCN5A Q14524 8/20 0.76
CSF1R P07333 8/20 0.69
MEN1 O00255 1/20 0.54
GAA P10253 1/20 0.54
SLC2A1 P11166 1/20 0.54
KMT2A Q03164 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910730 0.94 KCNH2 (0.85) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2904648 0.94 CSF1R (0.79) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2907777 0.94 KCNH2 (0.67) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2910626 0.92 KCNH2 (0.74) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2913359 0.91 CSF1R (0.66) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2911256 0.91 KCNH2 (0.76) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2912359 0.91 CSF1R (0.63) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2913869 0.90 CSF1R (0.86) KCNH2SCN5ACSF1R
SCHEMBL2911044 0.89 CSF1R (0.69) KCNH2SCN5ACSF1RMEN1GAA
SCHEMBL2911029 0.88 CSF1R (0.84) KCNH2SCN5ACSF1RMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed